I. Basic Information (API Foreign Trade Version)
English: Vibegron
Chinese: 维贝格龙
CAS No.: 1000307-35-0
Molecular Formula: C₂₄H₂₉N₅O₄
Molecular Weight: 451.52
Appearance: White to off-white powder
Type: Highly selective β3 adrenergic receptor agonist
II. Actions and Uses
For overactive bladder (OAB)
Relieves: Urinary frequency, urgency, and incontinence
Advantages:
Minimally invasive cardiovascular effects
Not extensively metabolized by CYP3A4, resulting in fewer drug interactions
Superior safety and tolerability compared to traditional anticholinergic drugs