Upadacitinib

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Selling leads
Upadacitinib
Posting date : Feb 25, 2026
Membership
Free Member Scince Jul 07, 2025
FOB Price
$243.5
Min. Order Quantity
10g
Supply Abillity
Stock
Port
Ningbo
Payment Terms
T/T 100%
Package
1g,10g,20g,
Keyword :
Category
Contact
Lunar
Selling Leads Detail
Company Info
 
Quick Detail
Place of Origin
China [CN]
Brand Name
Jinlan
HS-CODE
-
Package & Delivery Lead Time
Package
1g,10g,20g,
Detailed Description
CAS No.:1310726-60-7
Molecular Formula:C₁₇H₁₉F₃N₆O
Molecular Weight380.37

Characteristic

  • Appearance:White to off-white powder
  • Solubility:Slightly soluble in water, soluble in organic solvents
  • Storage:Sealed, dry, protected from light

Pharmacological Category

Selective JAK1 inhibitor (Janus kinase 1 inhibitor)
Immunomodulator / Anti-inflammatory agent

Mechanism of Action

  • Selectively inhibits JAK1
  • Blocks downstream signaling of multiple pro-inflammatory cytokines
  • Reduces inflammation, joint damage, and disease activity

Indications

  • Rheumatoid arthritis
  • Psoriatic arthritis
  • Ankylosing spondylitis
  • Atopic dermatitis
  • Ulcerative colitis
  • Crohn’s disease

Key Features

  • Oral, once-daily administration
  • High selectivity for JAK1
  • Broad efficacy across multiple immune-mediated inflammatory diseases

Main Adverse Reactions

  • Upper respiratory tract infections
  • Nausea
  • Increased liver enzymes
  • Lipid elevation
  • Headache

Contraindications

  • Hypersensitivity to upadacitinib or any excipient
  • Active severe infections

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